Intramolecular palladium mediated π-allyl cyclisation of bis-Cbz- and bis-Boc-protected guanidines

Zainab Al-Shuhaib, Henning Böckemeier, Lawrence Coghlan, Elina Dörksen, Iestyn V. Jones, Patrick J. Murphy, Robert J. Nash, James M. Page

Research output: Contribution to journalArticlepeer-review

3 Citations (SciVal)

Abstract

The Pd-mediated π-allyl cyclisation of bis-Cbz- and bis-Boc-protected guanidines 4 and 14b led to the formation of five- and six-membered heterocycles 5 and 17 in high yields.
Original languageEnglish
Pages (from-to)6716-6718
JournalTetrahedron Letters
Volume54
Issue number49
Early online date27 Sept 2013
DOIs
Publication statusPublished - 04 Dec 2013

Keywords

  • guanidine
  • palladium allylation
  • heterocyclisation
  • intramolecular cyclisation

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